SCHEMBL21546809

SCHEMBL21546809

N#Cc1cccc(-c2cc(-n3c4ccccc4c4cc(-c5ccc(-c6ccccc6)nc5)ccc43)c(C#N)c(-n3c4ccccc4c4cc(-c5ccc(-c6ccccc6)nc5)ccc43)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRA3 P34903 2/20 0.41
GABRA1 P14867 1/20 0.41
ALDH1A3 P47895 1/20 0.40
KDM1A O60341 1/20 0.38
MAP4K4 O95819 1/20 0.37
CYP11B1 P15538 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21546804 0.97 GABRG2 (0.44) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21414307 0.95 GABRA1 (0.35) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21546802 0.94 GABRG2 (0.41) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21546803 0.91 GABRG2 (0.44) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22760928 0.91 GABRG2 (0.37) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21547024 0.89 GABRG2 (0.39) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21546779 0.89 GABRG2 (0.42) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22760925 0.89 GABRG2 (0.42) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL21414308 0.89 GABRG2 (0.35) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL19909400 0.89 ALDH1A3 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3478793-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2019-11-06 EP disclosed