SCHEMBL21550130

SCHEMBL21550130

Cn1nc(Cl)c(CNC(=O)OC(C)(C)C)cc1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.41
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41
KDM4A O75164 1/20 0.39
GFER P55789 1/20 0.39
HDAC10 Q969S8 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
IDO1 P14902 2/20 0.37
PRMT5 O14744 2/20 0.36
WDR77 Q9BQA1 2/20 0.36
GAA P10253 1/20 0.36
STK17B O94768 1/20 0.36
STK17A Q9UEE5 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1B Q00975 1/20 0.36
CACNA1C Q13936 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8275252 0.76 KDM4A (0.43) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL20157969 0.74 TRPA1 (0.40) KDM4ELMNAATML3MBTL1GAA
SCHEMBL20157341 0.74 KDM4E (0.40) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL20157285 0.74 HDAC10 (0.40) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL13881841 0.72 AAK1 (0.43) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL28712496 0.70 LMNA (0.44) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL19782521 0.70 POLB (0.45) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL13881875 0.70 STK17B (0.46) POLBMAPK1ATMKDM4AGFER
SCHEMBL21425585 0.70 BRD4 (0.42) KDM4ELMNAPOLBMAPK1ATM
SCHEMBL16532758 0.70 GAA (0.48) KDM4ELMNAKDM4AL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed