SCHEMBL21553675

SCHEMBL21553675

CC(=O)NC(CSCC(N)=O)C(=O)NCC(N)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
ALDH1A1 P00352 2/20 0.36
OPRM1 P35372 1/20 0.36
SIRT6 Q8N6T7 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
KDM4E B2RXH2 1/20 0.33
THRB P10828 1/20 0.33
ALOX15 P16050 1/20 0.33
NFKB1 P19838 1/20 0.33
PTGS2 P35354 1/20 0.33
THPO P40225 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19277912 0.83 MAPT (0.38) MAPTALDH1A1KDM4ETHRBALOX15
SCHEMBL30493611 0.83 GNPAT (0.39) MAPTALDH1A1OPRM1SIRT6SIRT1
SCHEMBL27263098 0.82 ACE (0.35) ALDH1A1THRBFCER2TLR2
SCHEMBL30493797 0.80 SIRT6 (0.42) MAPTALDH1A1OPRM1SIRT6SIRT1
SCHEMBL24013206 0.80 FCER2 (0.40) SCN9AFCER2GLO1
SCHEMBL30493695 0.80 OPRM1 (0.38) MAPTALDH1A1OPRM1SIRT6SIRT1
SCHEMBL24899392 0.79 ACE (0.33) ALDH1A1OPRM1THRBFCER2TLR2
SCHEMBL18862364 0.78 MAPT (0.53) MAPTALDH1A1OPRM1SIRT6SIRT1
SCHEMBL23960483 0.77
SCHEMBL14008029 0.77 ALDH1A1 (0.55) MAPTALDH1A1OPRM1SMN1; SMN2CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970390-B1 MACROCYCLIC INHIBITORS OF THE PD-1/PD-L1 AND CD80(B7-1)/PD-L1 PROTEIN/PROTEIN INTERACTIONS BRISTOL MYERS SQUIBB CO (US) 2019-11-06 EP disclosed