SCHEMBL21557598

SCHEMBL21557598

c1ccc(-c2ccc3c(c2)CNC3)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
SYK P43405 1/20 0.44
KDM4E B2RXH2 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
CCR1 P32246 1/20 0.43
CCR5 P51681 1/20 0.43
CCR8 P51685 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
PDK2 Q15119 1/20 0.42
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41
PI4KA P42356 1/20 0.41
PIK3CG P48736 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833268 0.87 ASIC3 (0.49) HTR1AHTR7SYKASIC3
SCHEMBL1010747 0.87 ASIC3 (0.56) HTR1AHTR7SYKPIM1PIM3
SCHEMBL1011236 0.87 ASIC3 (0.49) HTR1AHTR7SYKASIC3
SCHEMBL31070452 0.81 KDM4E (0.39) HTR1AHTR7SYKKDM4ELMNA
SCHEMBL23351094 0.77 CYP11B1 (0.47) HTR1AHTR7KDM4ELMNACYP1A2
SCHEMBL4024459 0.77 CYP11B1 (0.51) HTR1AHTR7KDM4ELMNACYP1A2
SCHEMBL4025451 0.76 CYP11B1 (0.50) HTR1AHTR7KDM4ELMNACYP1A2
SCHEMBL21557592 0.75 PDK2 (0.40) HTR1AHTR7KDM4ELMNACYP1A2
SCHEMBL6130756 0.75 PDK2 (0.51) HTR1AHTR7KDM4ELMNACYP1A2
SCHEMBL20599454 0.74 NTRK2 (0.65) PDK2CYP2A6PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3566749-A1 THIAZOLE DERIVATIVE AND APPLICATIONS THEREOF Medshine Discovery Inc. (CN) 2019-11-13 EP disclosed