SCHEMBL21560180

SCHEMBL21560180

Cc1ccc(-c2nc(CC(=O)NC(c3ccc(Cl)cc3)C(O)O)cs2)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
LMNA P02545 3/20 0.48
CNR2 P34972 1/20 0.47
SHMT1 P34896 5/20 0.47
SHMT2 P34897 3/20 0.47
TP53 P04637 4/20 0.46
ALDH1A1 P00352 2/20 0.46
THRB P10828 1/20 0.45
GFER P55789 1/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21560010 0.89 KDM4E (0.54) MAPTLMNASHMT1SHMT2TP53
SCHEMBL20256000 0.85 SHMT1 (0.52) MAPTLMNACNR2SHMT1SHMT2
SCHEMBL20255618 0.78 SHMT1 (0.72) MAPTLMNASHMT1SHMT2TP53
SCHEMBL21559996 0.78 SHMT1 (0.72) MAPTLMNASHMT1SHMT2TP53
SCHEMBL8240059 0.77 SHMT1 (0.60) MAPTLMNASHMT1SHMT2TP53
SCHEMBL20255559 0.77 SHMT2 (0.69) MAPTLMNASHMT1SHMT2ALDH1A1
SCHEMBL20255621 0.77 SHMT2 (0.69) MAPTLMNASHMT1SHMT2ALDH1A1
SCHEMBL20255951 0.76 SHMT1 (0.58) MAPTLMNASHMT1SHMT2TP53
SCHEMBL20255675 0.76 SHMT1 (0.58) MAPTLMNASHMT1SHMT2TP53
SCHEMBL20255891 0.76 SHMT1 (0.55) MAPTSHMT1SHMT2TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11091451-B2 SHMT inhibitors and uses thereof RAZE THERAPEUTICS, INC. (US) 2021-08-17 US disclosed
US-20190345119-A1 SHMT INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. 2019-11-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11091451-B2 SHMT inhibitors and uses thereof SHMT1, SHMT2, BHMT MAPT 1852/4885LMNA 4283/4885CNR2 4713/4885
US-20190345119-A1 SHMT INHIBITORS AND USES THEREOF SHMT1, SHMT2, BHMT MAPT 1852/4885LMNA 4283/4885CNR2 4713/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.