SCHEMBL2156359

SCHEMBL2156359

COC(=O)c1cc2[nH]c(Br)c(-c3ccccc3)c2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 8/20 0.40
RAB9A P51151 1/20 0.40
HPGD P15428 4/20 0.40
MAPT P10636 4/20 0.39
GAA P10253 2/20 0.39
PAK4 O96013 1/20 0.39
CSNK2A2 P19784 1/20 0.39
AKT1 P31749 1/20 0.39
PLK1 P53350 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
KDM4E B2RXH2 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
NR4A2 P43354 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2996447 0.88 ALDH1A1 (0.41) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2987902 0.86 LMNA (0.45) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2156447 0.80 RAF1 (0.40) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2986582 0.80 PTGS2 (0.42) LMNAALDH1A1RAB9AHPGDMAPT
SCHEMBL2863437 0.79 LMNA (0.38) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2868302 0.79 ALDH1A1 (0.40) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2157797 0.76 LMNA (0.37) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2993837 0.75 PAK4 (0.43) LMNAMEN1KMT2AALDH1A1RAB9A
SCHEMBL2156336 0.74 HTT (0.51) LMNAMEN1KMT2AALDH1A1HPGD
SCHEMBL2859156 0.73 ALDH1A1 (0.38) LMNAMEN1KMT2AALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7973026-B2 Thienopyrroles as antiviral agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2011-07-05 US disclosed
US-7659263-B2 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2010-02-09 US disclosed
US-7659263-B2 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2010-02-09 US disclosed
US-7659263-B2 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2010-02-09 US disclosed
US-20090105227-A1 Thienopyrroles As Antiviral Agents ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2009-04-23 US disclosed
EP-1881989-A1 THIENOPYRROLES AS ANTIVIRAL AGENTS Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2008-01-30 EP disclosed
WO-2006119975-A1 THIENOPYRROLES AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI SPA (IT) 2006-11-16 WO disclosed
US-20060167246-A1 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2006-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060167246-A1 Thienopyrrole compound and use thereof as HCV polymerase inhibitor TPMT, JAK2, GTF3C5 LMNA 4828/4885MEN1 4852/4885KMT2A 2063/4885
US-20090105227-A1 Thienopyrroles As Antiviral Agents ZC3HAV1, HAVCR2, ZC3HAV1L LMNA 4377/4885MEN1 4599/4885KMT2A 3202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.