SCHEMBL21574645

SCHEMBL21574645

C=CC(C=C)Cc1ccc(C(C)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
GRB2 P62993 1/20 0.33
MMP13 P45452 2/20 0.33
ACACB O00763 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PTPN1 P18031 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21075947 0.84 TAAR1 (0.45) NPC1RAB9AALDH1A1TAAR1
SCHEMBL18856419 0.80 TP53 (0.35) TP53TSHRGRB2MMP13ACACB
SCHEMBL18856426 0.73 TRPA1 (0.45) ESR1ESR2TAAR1
SCHEMBL12299036 0.71 TSHR (0.40) TSHRALDH1A1ESR1ESR2NR1H2
SCHEMBL22059353 0.70 TSHR (0.39) TP53TSHRGRB2ACACBALDH1A1
SCHEMBL1061707 0.70 EPHX1 (0.48) TAAR1SLC6A4
SCHEMBL11932056 0.70 TP53 (0.42) TP53TSHRNPC1RAB9AALDH1A1
SCHEMBL11932058 0.70 TAAR1 (0.37) TP53TSHRPTPN1ALDH1A1ESR1
SCHEMBL21076021 0.69 HTR2A (0.60) TP53TSHRALDH1A1TAAR1SLC6A4
SCHEMBL19143516 0.69 GRB2 (0.55) GRB2ACACBPTPN1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057951-B1 METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T JANSSEN PHARMACEUTICA NV (BE) 2019-11-20 EP disclosed