SCHEMBL18856419

SCHEMBL18856419

C=CC(Cc1ccc(C(C)(F)F)cc1)C(=C)C

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
GRB2 P62993 1/20 0.35
ACACB O00763 3/20 0.33
PTPN1 P18031 1/20 0.33
MMP13 P45452 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21574645 0.80 TP53 (0.41) TP53TSHRGRB2ACACBPTPN1
SCHEMBL21538871 0.75 HTR2A (0.55) TP53TSHR
SCHEMBL21076020 0.74 PPARG (0.38) TP53TSHR
SCHEMBL21574736 0.73 IDO1 (0.39)
SCHEMBL21573071 0.73 HRH3 (0.37) TP53TSHR
SCHEMBL19143516 0.69 GRB2 (0.55) GRB2ACACBPTPN1
SCHEMBL11932058 0.67 TAAR1 (0.37) TP53TSHRPTPN1
SCHEMBL24202494 0.66 CPA1 (0.41) MMP13
SCHEMBL1742369 0.66 EPHX2 (0.44) TSHR
SCHEMBL21075947 0.65 TAAR1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2909192-B1 METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T JANSSEN PHARMACEUTICA NV (BE) 2017-05-17 EP disclosed