SCHEMBL21574976

SCHEMBL21574976

CC(=O)NSc1ccc(CN(CCc2ccc(Br)cc2)C2CCNCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.39
SLC6A4 P31645 11/20 0.39
SLC6A3 Q01959 4/20 0.39
TACR1 P25103 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 1/20 0.36
MBTPS1 Q14703 1/20 0.36
CHIT1 Q13231 1/20 0.35
CHIA Q9BZP6 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17853346 0.82 PPARG (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL17838856 0.81 PPARG (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL21575105 0.80 TACR1 (0.42) SLC6A2SLC6A4SLC6A3TACR1MEN1
SCHEMBL548295 0.75 SLC6A4 (0.52) SLC6A2SLC6A4SLC6A3TACR1MEN1
SCHEMBL17853443 0.74 CA2 (0.44) SLC6A2SLC6A4SLC6A3TACR1CHIT1
Hydrochloric Acid SCHEMBL17838889 0.73 CA2 (0.43) SLC6A2SLC6A4SLC6A3TACR1CHIT1
SCHEMBL16097011 0.69 SLC6A2 (0.64) SLC6A2SLC6A4SLC6A3TACR1MEN1
SCHEMBL16825796 0.68 CHIA (0.53) SLC6A2SLC6A4SLC6A3CHIT1CHIA
SCHEMBL17838827 0.67 KMT2A (0.47) MEN1KMT2AALDH1A1CHIT1CHIA
SCHEMBL5583514 0.66 ABCB11 (0.48) SLC6A2SLC6A4SLC6A3KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233832-B1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS ONCOARENDI THERAPEUTICS SA (PL) 2019-11-20 EP disclosed