SCHEMBL2158751

SCHEMBL2158751

CC(C)N(C(=O)c1ccc(Cl)cc1Cl)c1csc(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.45
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
ALDH1A1 P00352 4/20 0.38
ALOX12 P18054 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
GAA P10253 1/20 0.37
FLT1 P17948 3/20 0.37
FLT4 P35916 3/20 0.37
KDR P35968 3/20 0.37
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157722 0.86 CYP3A4 (0.46) CYP3A4TSHRCASP1SMN1; SMN2SLC6A2
SCHEMBL2158295 0.81 CYP3A4 (0.41) CYP3A4TSHRCASP1SMN1; SMN2ALDH1A1
SCHEMBL2158071 0.78 HSD17B1 (0.43) CYP3A4TSHRSMN1; SMN2ALDH1A1NPC1
SCHEMBL1959495 0.75 TSHR (0.42) CYP3A4TSHRCASP1SMN1; SMN2SLC6A2
SCHEMBL6017639 0.73 TSHR (0.43) CYP3A4TSHRCASP1SMN1; SMN2SLC6A2
SCHEMBL1961039 0.72 FLT1 (0.39) CYP3A4SMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL6627206 0.71 PDK1 (0.44) CYP3A4TSHRCASP1SMN1; SMN2FLT1
SCHEMBL4159892 0.70 MAPT (0.45) CYP3A4SMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL2157949 0.69 POLB (0.45) ALDH1A1
SCHEMBL13270806 0.69 SMN1; SMN2 (0.41) CYP3A4TSHRCASP1SMN1; SMN2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985769-B2 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-26 US disclosed
US-20060142347-A1 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS (CANADA) INCORPORATED (CA) 2006-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060142347-A1 Compounds and methods for the treatment or prevention of Flavivirus infections HAVCR2, ZC3HAV1, MAVS CYP3A4 622/4885TSHR 4609/4885CASP1 64/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.