SCHEMBL21589799

SCHEMBL21589799

CCCCC1(CCCC)CSc2cc(O/C=C/C(=O)O)c(F)cc2N(c2ccccc2)C1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 1/20 0.33
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21589722 0.96 USP2 (0.30) LTB4R2USP2ALDH1A1POLBALOX15
SCHEMBL21589514 0.90 RORC (0.31)
SCHEMBL21589718 0.89 NR1H4 (0.36)
SCHEMBL21589626 0.87 RORC (0.30)
SCHEMBL21589772 0.85
SCHEMBL21589858 0.85
SCHEMBL23481680 0.85 PTGDR2 (0.35) TSHRHSD17B10
SCHEMBL21586028 0.85 DRD2 (0.33) USP2ALDH1A1POLBALOX15TSHR
SCHEMBL22476248 0.83 NR1H4 (0.32) LTB4R2
SCHEMBL21589790 0.83 SLC10A2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802504-B1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2023-01-18 EP disclosed
WO-2019234077-A1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2019-12-12 WO disclosed