SCHEMBL21589906

SCHEMBL21589906

COc1cc(-c2ccc(N(C)c3ccc(CN(C)C)cc3)cc2)ccc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.49
HTR7 P34969 4/20 0.48
TAAR1 Q96RJ0 2/20 0.44
TNKS O95271 2/20 0.43
BRD4 O60885 2/20 0.42
BRD9 Q9H8M2 2/20 0.42
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR1E P28566 1/20 0.38
HTR2B P41595 1/20 0.38
HTR3A P46098 1/20 0.38
HTR5A P47898 1/20 0.38
HTR6 P50406 1/20 0.38
PARP1 P09874 1/20 0.38
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31207326 0.84 HRH3 (0.47) HRH3HTR7TAAR1TNKSBRD4
SCHEMBL23630637 0.84 HRH3 (0.47) HRH3HTR7TAAR1TNKSBRD4
SCHEMBL17117158 0.76 ALDH1A1 (0.54)
SCHEMBL9440147 0.74 ALDH1A1 (0.56)
SCHEMBL13335119 0.70 ALDH1A1 (0.48) TNKSACHE
SCHEMBL13681448 0.70 CSF1R (0.43) HTR7
SCHEMBL12679031 0.70 HRH3 (1.00) HRH3TAAR1TNKSBRD4BRD9
SCHEMBL14426480 0.70 HTR7 (0.60) HRH3HTR7HTR1AHTR1DHTR1B
SCHEMBL31207322 0.69 HRH3 (0.46) HRH3HTR7TAAR1
SCHEMBL23630646 0.69 HRH3 (0.46) HRH3HTR7TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019234405-A1 COMPOUNDS USEFUL IN THE TREATMENT OF DISORDERS ASSOCIATED WITH MUTANT RAS OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2019-12-12 WO disclosed