SCHEMBL21590337

SCHEMBL21590337

CNC(=O)c1ncccc1CCCOC

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
GCK P35557 3/20 0.42
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 4/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
HTT P42858 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 2/20 0.38
GAA P10253 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29289961 0.82 PARP1 (0.49) PARP1KDM4EALDH1A1CYP1A2MAPT
SCHEMBL27601273 0.81 PARP1 (0.48) PARP1KDM4EALDH1A1L3MBTL1LMNA
SCHEMBL15966073 0.80 PARP1 (0.52) PARP1KDM4EALDH1A1L3MBTL1CYP1A2
SCHEMBL2160307 0.79 PARP1 (0.51) PARP1KDM4EALDH1A1L3MBTL1CYP1A2
SCHEMBL19539578 0.78 ALDH1A1 (0.47) PARP1KDM4EALDH1A1HTTTDP1
SCHEMBL7218347 0.77 PARP1 (0.50) PARP1KDM4EALDH1A1L3MBTL1POLB
SCHEMBL28019213 0.77 PKM (0.45) GCKKDM4EALDH1A1L3MBTL1HTT
SCHEMBL21590248 0.76 TSHR (0.49) KDM4EALDH1A1L3MBTL1HTTPOLB
SCHEMBL22018876 0.76 KDM4E (0.58) KDM4EALDH1A1L3MBTL1CYP1A2MAPT
SCHEMBL28805406 0.75 KDM4E (0.41) PARP1KDM4EALDH1A1L3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed