SCHEMBL21591751

SCHEMBL21591751

Nc1ncccc1Cc1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.47
MPO P05164 1/20 0.47
BACE1 P56817 2/20 0.46
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
CYP2A6 P11509 1/20 0.44
HTT P42858 1/20 0.44
PNP P00491 1/20 0.44
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
MMP2 P08253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30969090 0.86 BACE1 (0.43) CHRNA7MPOBACE1CYP11B1CYP11B2
SCHEMBL2259723 0.83 LTA4H (0.53) BACE1
SCHEMBL9694096 0.83 MPO (0.48) CHRNA7MPOCYP11B1CYP11B2CYP1A2
Ammonia Solution, Strong SCHEMBL4936578 0.82 BACE1 (0.61) BACE1CYP11B1CYP11B2CYP1A2CYP2A6
SCHEMBL4418570 0.80 HTT (0.49) CHRNA7MPOCYP11B1CYP11B2CYP1A2
Hydrochloric Acid SCHEMBL11398017 0.79 HTT (0.47) CHRNA7MPOCYP11B1CYP11B2CYP1A2
SCHEMBL27836688 0.79 HTT (0.51) CHRNA7CYP11B1CYP11B2CYP1A2CYP2D6
SCHEMBL3962268 0.78 DHFR (0.60)
SCHEMBL30612271 0.77 CHRNA7 (0.46) CHRNA7MPOCYP11B1CYP11B2CYP1A2
SCHEMBL9665011 0.77 CHRNA7 (0.46) CHRNA7MPOCYP11B1CYP11B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3807273-A1 AZAINDOLE DERIVATIVES AS RHO- KINASE INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2021-04-21 EP claimed
WO-2019238628-A1 AZAINDOLE DERIVATIVES AS RHO- KINASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2019-12-19 WO claimed