SCHEMBL21593358

SCHEMBL21593358

COc1cc(Br)cc(CCN(C=O)CC#N)c1C

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.33
ERN1 O75460 1/20 0.33
HTR2A P28223 1/20 0.33
ELANE P08246 1/20 0.32
PYCR1 P32322 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21593329 0.85 ALDH1A1 (0.38) GAAERN1HTR2AALDH1A1CYP1A2
SCHEMBL31689789 0.65 MC4R (0.40) HTR2AALDH1A1
SCHEMBL28855352 0.64 PDE4A (0.47) GAAERN1
SCHEMBL15525407 0.63 NQO2 (0.47) ERN1ALDH1A1
SCHEMBL16475647 0.62 ERN1 (0.68) ERN1ALDH1A1CYP1A2CYP2C19
SCHEMBL24169418 0.59 KMT2A (0.38) GAAERN1HTR2AALDH1A1
SCHEMBL27933933 0.59 CYP1A2 (0.41) GAAERN1HTR2AALDH1A1CYP1A2
SCHEMBL7617001 0.59
SCHEMBL6672627 0.58 NQO2 (0.47) ERN1ALDH1A1
SCHEMBL12561405 0.58 ALOX15 (0.50) ERN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238424-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2019-12-19 WO disclosed