SCHEMBL21596943

SCHEMBL21596943

COc1c(Br)ccc2noc(N)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 3/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
HSD17B10 Q99714 3/20 0.32
USP2 O75604 2/20 0.32
ALOX15 P16050 2/20 0.32
APAF1 O14727 1/20 0.32
TDP2 O95551 1/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
BRCA1 P38398 1/20 0.32
CASP7 P55210 1/20 0.32
CA4 P22748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596939 0.74 PTGS1 (0.30)
SCHEMBL29652416 0.73 KDR (0.37) NQO2MEN1KMT2AKDM4ERAB9A
SCHEMBL21596851 0.73 KDR (0.37) NQO2MEN1KMT2AKDM4ERAB9A
SCHEMBL24344354 0.70 NQO2 (0.41) NQO2MEN1KMT2AMAPTALOX5AP
SCHEMBL30770136 0.70 TDP2 (0.45) NQO2ALOX5APFEN1TDP2
SCHEMBL21596942 0.69 BACE1 (0.40) CA4
SCHEMBL21596932 0.69 DCPS (0.51) NQO2MEN1KMT2AKDM4EALDH1A1
SCHEMBL21596930 0.67 NQO2 (0.41) NQO2MEN1KMT2AKDM4ERAB9A
SCHEMBL1519286 0.66 ALOX5AP (0.40) NQO2MEN1KMT2ARAB9AMAPT
SCHEMBL29514108 0.66 ALOX5AP (0.40) NQO2MEN1KMT2ARAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810602-A1 COMPOUNDS CTXT Pty Limited (AU) 2021-04-28 EP disclosed
WO-2019243491-A1 COMPOUNDS CTXT PTY LIMITED (AU) 2019-12-26 WO disclosed