SCHEMBL21609199

SCHEMBL21609199

Nc1cc(F)c(Cl)nc1O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
KHK P50053 1/20 0.36
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
SLC9A1 P19634 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8235252 0.79 KEAP1 (0.47) KEAP1NFE2L2KHKTDP1ALDH1A1
SCHEMBL29829949 0.77 KEAP1 (0.41) KEAP1NFE2L2KHKTDP1ALDH1A1
SCHEMBL23620152 0.77 KEAP1 (0.41) KEAP1NFE2L2KHKTDP1ALDH1A1
SCHEMBL26712680 0.74 KEAP1 (0.38) KEAP1NFE2L2KHKTDP1
SCHEMBL12608076 0.74 KEAP1 (0.38) KEAP1NFE2L2KHKTDP1
SCHEMBL31453136 0.74 KEAP1 (0.38) KEAP1NFE2L2KHKTDP1
SCHEMBL30296610 0.74 KEAP1 (0.38) KEAP1NFE2L2KHKTDP1
SCHEMBL16101278 0.72 KEAP1 (0.55) KEAP1NFE2L2KHKTDP1ALDH1A1
SCHEMBL29260193 0.70 KEAP1 (0.56) KEAP1NFE2L2KHKTDP1
SCHEMBL29140679 0.70 PTK2 (0.44) ALDH1A1HPGDALOX15ALOX12MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019243303-A1 PYRIDINYL AND PYRAZINYL-(AZA)INDOLSULFONAMIDES UCB PHARMA GMBH (DE) 2019-12-26 WO disclosed