SCHEMBL21621709

SCHEMBL21621709

Cc1c(CO)cccc1-n1c(C)nc(CO)c1C

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.40
CD274 Q9NZQ7 2/20 0.40
GAA P10253 1/20 0.34
HCAR1 Q9BXC0 1/20 0.33
POLB P06746 1/20 0.33
SETDB1 Q15047 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
P2RX7 Q99572 1/20 0.32
TP53 P04637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708065 0.78 TSHR (0.59) PDCD1CD274POLBTP53KDM4E
SCHEMBL11166064 0.76 PDCD1 (0.47) PDCD1CD274GAAPOLBMEN1
SCHEMBL21621663 0.74 ALDH1A1 (0.41) PDCD1CD274HCAR1MEN1KMT2A
SCHEMBL21621715 0.74 NOTUM (0.50) PDCD1CD274P2RX7TP53ALDH1A1
SCHEMBL10153084 0.73 MAPK1 (0.47) HCAR1MEN1KMT2AALDH1A1TSHR
SCHEMBL1708275 0.70 BMI1 (0.37) HCAR1ALDH1A1TSHR
SCHEMBL9454981 0.69 PDCD1 (0.47) PDCD1CD274GAAKMT2ATP53
SCHEMBL1708353 0.69 L3MBTL1 (0.38) PDCD1CD274ALDH1A1TSHR
SCHEMBL10153088 0.69 SORD (0.41) PDCD1CD274MEN1KMT2AKDM4E
SCHEMBL6424004 0.69 PDCD1 (0.64) PDCD1CD274MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020011246-A1 BENZENE RING-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 广州丹康医药生物有限公司 2020-01-16 WO disclosed