SCHEMBL21628148

SCHEMBL21628148

Cc1nn(CC(=O)NN)c(C)c1Br

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
PKM P14618 2/20 0.51
RECQL P46063 1/20 0.51
APAF1 O14727 1/20 0.50
HTT P42858 3/20 0.49
GAA P10253 3/20 0.44
NPSR1 Q6W5P4 2/20 0.43
AGTR1 P30556 1/20 0.43
LMNA P02545 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15229912 0.85 APAF1 (0.55) KDM4EALDH1A1PKMAPAF1HTT
SCHEMBL15229836 0.81 HTT (0.62) KDM4EALDH1A1PKMAPAF1HTT
SCHEMBL15229985 0.80 APAF1 (0.47) KDM4EALDH1A1PKMAPAF1HTT
SCHEMBL15231004 0.79 APAF1 (0.56) ALDH1A1APAF1HTTGAANPSR1
SCHEMBL3585241 0.79 ALDH1A1 (0.67) ALDH1A1APAF1HTTGAALMNA
Ethane SCHEMBL11828584 0.77 ALDH1A1 (0.65) ALDH1A1APAF1HTTGAALMNA
SCHEMBL15230043 0.75 APAF1 (0.51) KDM4EALDH1A1PKMAPAF1HTT
SCHEMBL21654553 0.74 GAA (0.61) ALDH1A1RECQLAPAF1HTTGAA
SCHEMBL15230436 0.73 APAF1 (0.50) ALDH1A1PKMAPAF1HTTLMNA
SCHEMBL11831505 0.71 RAB9A (0.43) ALDH1A1APAF1HTTLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11149033-B2 Heteroaryl compound, enantiomer, diastereomer or pharmaceutically acceptable salt thereof, and antiviral composition containing same as active ingredient INSTITUT PASTEUR KOREA (KR) 2021-10-19 US disclosed
US-11149033-B2 Heteroaryl compound, enantiomer, diastereomer or pharmaceutically acceptable salt thereof, and antiviral composition containing same as active ingredient INSTITUT PASTEUR KOREA (KR) 2021-10-19 US disclosed
US-20200031816-A1 NOVEL HETEROARYL COMPOUND, ENANTIOMER, DIASTEREOMER OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND ANTIVIRAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT ST PHARM CO., LTD. (KR) 2020-01-30 US disclosed
US-20200031816-A1 NOVEL HETEROARYL COMPOUND, ENANTIOMER, DIASTEREOMER OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND ANTIVIRAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT ST PHARM CO., LTD. (KR) 2020-01-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200031816-A1 NOVEL HETEROARYL COMPOUND, ENANTIOMER, DIASTEREOMER OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND ANTIVIRAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT ZC3HAV1, ZC3HAV1L, HAVCR2 KDM4E 3325/4885ALDH1A1 980/4885PKM 3287/4885
US-11149033-B2 Heteroaryl compound, enantiomer, diastereomer or pharmaceutically acceptable salt thereof, and antiviral composition containing same as active ingredient ZC3HAV1, ZC3HAV1L, HAVCR2 KDM4E 3277/4885ALDH1A1 839/4885PKM 3118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.