SCHEMBL2164772

SCHEMBL2164772

O=C1C=C(c2ccccc2)/C(=C\c2ccccc2)O1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 5/20 0.49
HPGD P15428 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
MAPT P10636 3/20 0.47
MITF O75030 1/20 0.47
LMNA P02545 1/20 0.47
NTSR1 P30989 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
STK17B O94768 1/20 0.45
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
BACE1 P56817 1/20 0.38
PNLIP P16233 1/20 0.38
ACHE P22303 1/20 0.38
DAPK3 O43293 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2164768 1.00 KDM4E (0.49) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL2164776 1.00 KDM4E (0.49) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL30674009 0.85 ALOX5 (0.46) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL30674001 0.85 PLCG2 (0.56) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL30674010 0.85 MAPT (0.41) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL13492163 0.85 MAOB (0.44) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL2167197 0.83 KDM4E (0.41) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL2315391 0.83 MAPT (0.40) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL2315392 0.83 MAPT (0.40) KDM4EALDH1A1HPGDL3MBTL1TDP1
SCHEMBL2165995 0.83 MAPT (0.40) KDM4EALDH1A1HPGDL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350036-B1 METHYLENE FURANONE DERIVATIVES AND USE OF SAID DERIVATIVES AS A PHOTOPROTECTING OR ANTIOXIDANT OR DEPIGMENTATION AGENT IN COSMETIC OR DERMATOLOGICAL COMPOSITIONS PIERRE FABRE DERMO COSMÉTIQUE (FR) 2015-04-15 EP disclosed
US-8563548-B2 Methylene furanone derivatives and use of said derivatives as a photoprotecting or antioxidant or depigmentation agent in cosmetic or dermatological compositions PIERRE FABRE DERMO-COSMETIQUE (FR) 2013-10-22 US disclosed
EP-2350036-A1 METHYLENE FURANONE DERIVATIVES AND USE OF SAID DERIVATIVES AS A PHOTOPROTECTING OR ANTIOXIDANT OR DEPIGMENTATION AGENT IN COSMETIC OR DERMATOLOGICAL COMPOSITIONS Pierre Fabre Dermo-Cosmétique (FR) 2011-08-03 EP disclosed
US-20110184059-A1 METHYLENE FURANONE DERIVATIVES AND USE OF SAID DERIVATIVES AS A PHOTOPROTECTING OR ANTIOXIDANT OR DEPIGMENTATION AGENT IN COSMETIC OR DERMATOLOGICAL COMPOSITIONS PIERRE FABRE DERMO-COSMETIQUE (FR) 2011-07-28 US disclosed
WO-2010034827-A1 METHYLENE FURANONE DERIVATIVES AND USE OF SAID DERIVATIVES AS A PHOTOPROTECTING OR ANTIOXIDANT OR DEPIGMENTATION AGENT IN COSMETIC OR DERMATOLOGICAL COMPOSITIONS PIERRE FABRE DERMO-COSMETIQUE (FR) 2010-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110184059-A1 METHYLENE FURANONE DERIVATIVES AND USE OF SAID DERIVATIVES AS A PHOTOPROTECTING OR ANTIOXIDANT OR DEPIGMENTATION AGENT IN COSMETIC OR DERMATOLOGICAL COMPOSITIONS NQO1, ESD, DHPS KDM4E 243/4885ALDH1A1 147/4885HPGD 138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.