SCHEMBL2165685

SCHEMBL2165685

N#Cc1nc(Cl)ccc1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.37
CSNK1A1 P48729 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
POLB P06746 1/20 0.33
IDO1 P14902 1/20 0.33
GAA P10253 1/20 0.33
KHK P50053 1/20 0.32
USP8 P40818 3/20 0.32
USP7 Q93009 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
ADORA2B P29275 1/20 0.32
USP47 Q96K76 1/20 0.32
ERBB2 P04626 1/20 0.32
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7108696 0.77 KDM4E (0.39) KDM4EALDH1A1POLBGAAUSP8
SCHEMBL30450356 0.77 KDM4E (0.39) KDM4EALDH1A1POLBGAAUSP8
SCHEMBL2708620 0.76 RPS6KA5 (0.39) CSNK1A1CLK4KDM4EALDH1A1POLB
Ammonia Solution, Strong SCHEMBL28870434 0.76 KDM4E (0.38) KDM4EALDH1A1POLBGAAUSP8
SCHEMBL15431202 0.75 GRM5 (0.34) PIK3CDSIRT2IDO1
SCHEMBL28457319 0.75 SIRT2 (0.32) PIK3CDSIRT2IDO1
SCHEMBL10960474 0.74 KDM4E (0.33) SIRT2KDM4EALDH1A1POLBGAA
SCHEMBL21816291 0.74 GRM5 (0.46) PIK3CDCLK4KDM4EALDH1A1POLB
SCHEMBL21248120 0.74 PIK3CD (0.33) PIK3CDKHKUSP8USP7ADORA2A
SCHEMBL12665887 0.74 PIK3CD (0.33) PIK3CDKDM4EUSP8ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122055367-A 5-Oxo-4, 5-dihydroimidazo [1,5-a ] quinazoline compounds as PI3K [ alpha ] inhibitors 皮卡维森治疗学股份有限公司 2026-05-15 CN disclosed
US-12617789-B2 Small molecular inhibitors of NF-κb inducing kinase JANSSEN PHARMACEUTICA NV (BE) 2026-05-05 US disclosed
US-20250270213-A1 PI3Ka INHIBITORS PIKAVATION THERAPEUTICS, INC. 2025-08-28 US disclosed
WO-2025085474-A1 5-OXO-4,5-DIHYDROIMIDAZO[1,5-A]QUINAZOLINE COMPOUNDS AS PI3K[ALPHA] INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2025-04-24 WO disclosed
CN-114269720-B Acetyl-coa synthetase short chain2(ACSS2) Small molecule inhibitors of (a) 库拉德夫制药私人有限公司 2025-03-28 CN disclosed
EP-4522608-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2025-03-19 EP disclosed
CN-119654321-A PI3K alpha inhibitors 突触活化疗法股份有限公司 2025-03-18 CN disclosed
CN-119546602-A Pyrrolidone derivatives as inhibitors of nfkb-induced kinase 詹森药业有限公司 2025-02-28 CN disclosed
EP-4511373-A1 PI3K? INHIBITORS Synnovation Therapeutics, Inc. (US) 2025-02-26 EP disclosed
EP-4482831-A1 NOVEL BICYCLIC COMPOUNDS AS RAD51 INHIBITORS Satya Therapeutics, Inc. (US) 2025-01-01 EP disclosed
CN-1349412-A Cyclic therapy using cyclic urea and cyclic amide derivatives AMERICAN HOME PROD (US) 2002-05-15 CN disclosed
US-6369056-B1 AGONISTS AND ANTAGONISTS OF THE PROGESTERONE RECEPTOR; CONTRACEPTIVES; 6-(3-CHLOROPHENYL)-4,4-DIMETHYL-1,4-DIHYDRO -3-OXA-1,8-DIAZA-NAPHTHALENE-2-ONE AND 6-CHLORO-4,4-DIMETHYL-1,4-DIHYDRO-3-OXA-1,5-DIAZA-NAPHTHALEN-2-ONE AMERICAN HOME PRODUCTS CORPORATION 2002-04-09 US disclosed
EP-1173208-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2002-01-23 EP disclosed
EP-1173443-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES American Home Products Corporation (US) 2002-01-23 EP disclosed
WO-2000066103-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed
WO-2000066592-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed
US-5639753-A CONTROLLING INSECTS IN AGRICULTURE CROPS FMC CORPORATION (US) 1997-06-17 US disclosed
US-5532367-A LARVICIDES FMC CORPORATION (US) 1996-07-02 US disclosed
US-5521190-A USEFUL AGAINST TOBACCO BUDWORM FMC CORPORATION (US) 1996-05-28 US disclosed
WO-1994027439-A1 INSECTICIDAL PTERIDINES AND 8-DEAZAPTERIDINES FMC CORPORATION (US) 1994-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12617789-B2 Small molecular inhibitors of NF-κb inducing kinase IRAK3, IKBKB, IKBKG PIK3CD 511/4885CSNK1A1 301/4885CLK4 1068/4885
US-20250270213-A1 PI3Ka INHIBITORS PIK3CA, PIK3C2A, PIK3R5 PIK3CD 4/4885CSNK1A1 358/4885CLK4 3046/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.