SCHEMBL21657749

SCHEMBL21657749

FC(F)(F)c1ccccc1-n1cc2ccc(Br)cc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.39
AADAT Q8N5Z0 1/20 0.39
MAPT P10636 4/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 2/20 0.37
LMNA P02545 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37
PMP22 Q01453 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
POLB P06746 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23320550 0.75 NPC1 (0.57) MAPTALDH1A1MEN1LMNAKMT2A
SCHEMBL29090390 0.74 NOTUM (0.40) PTGESMAPTMEN1LMNAKMT2A
SCHEMBL23320407 0.71 FBP1 (0.38) MAPTMEN1LMNAKMT2AHTT
SCHEMBL17441671 0.70 MAPT (0.45) MAPTALDH1A1MEN1LMNAKMT2A
SCHEMBL16112325 0.68 ALDH1A1 (0.45) AADATMAPTALDH1A1MEN1LMNA
SCHEMBL21484056 0.68 NOTUM (0.37) MAPTALDH1A1MEN1LMNAKMT2A
SCHEMBL26529726 0.67 MAPT (0.41) PTGESMAPTALDH1A1MEN1LMNA
SCHEMBL29969276 0.67 MAPT (0.44) MAPTALDH1A1MEN1LMNAKMT2A
SCHEMBL17440801 0.67 IRAK4 (0.39) MAPTMEN1LMNAKMT2ACYP1A2
SCHEMBL29968961 0.67 MAPT (0.42) MAPTALDH1A1MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020021024-A1 SUBSTITUTED BICYCLIC COMPOUNDS AS MODULATORS OF THE ARYL HYDROCARBON RECEPTOR (AHR) PHENEX PHARMACEUTICALS AG (DE) 2020-01-30 WO disclosed