Deferoxamine

Deferoxamine

SCHEMBL2165915

CC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCNC(=O)CCC(=O)N(O)CCCCCN.CS(=O)(=O)O.Cl.[Fe]

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Deferoxamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.95
LMNA P02545 1/20 0.95
GAA P10253 1/20 0.95
SMN1; SMN2 Q16637 1/20 0.95
KDM4A O75164 11/20 0.88
HIF1A Q16665 1/20 0.88
TET2 Q6N021 1/20 0.88
DOHH Q9BU89 1/20 0.88
SLC6A5 Q9Y345 2/20 0.41
PAOX Q6QHF9 2/20 0.41
KDM4C Q9H3R0 10/20 0.39
CASP2 P42575 1/20 0.34
KDM5A P29375 1/20 0.33
KDM7A Q6ZMT4 1/20 0.33
PHF8 Q9UPP1 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Deferoxamine SCHEMBL3953046 0.99 KDM4E (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL7715593 0.97 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL1699778 0.97 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL119982 0.97 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
SCHEMBL30036991 0.97 KDM4E (1.00) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL9351925 0.96 KDM4E (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL1034134 0.95 KDM4E (0.95) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL1509901 0.95 KDM4A (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL3115584 0.95 KDM4A (0.97) KDM4ELMNAGAASMN1; SMN2KDM4A
Deferoxamine SCHEMBL9555338 0.94 KDM4E (0.93) KDM4ELMNAGAASMN1; SMN2KDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385933-B1 CULTURE MEDIUM FOR CELL GROWTH AND TRANSFECTION LIFE TECHNOLOGIES CORP (US) 2012-07-11 EP disclosed
EP-2351827-A1 Culture medium for cell growth and transfection Life Technologies Corporation (US) 2011-08-03 EP disclosed
US-20110183375-A1 METAL BINDING COMPOUNDS AND THEIR USE IN CELL CULTURE MEDIUM COMPOSITIONS Life Technologies Corporation (US) 2011-07-28 US disclosed
US-20080286868-A1 METAL BINDING COMPOUNDS AND THEIR USE IN CELL CULTURE MEDIUM COMPOSITIONS INVITROGEN CORPORATION (US) 2008-11-20 US disclosed
US-6767741-B1 THE COMPOSITIONS OBVIATE THE NEED FOR NATURALLY DERIVED METAL-BINDING PROTEINS, SUCH AS TRANSFERRIN AND CERULOPLASMIN, WHICH MAY CONTAIN BLOOD-BORNE PATHOGENS INVITROGEN CORPORATION 2004-07-27 US disclosed