SCHEMBL21661355

SCHEMBL21661355

CCC(=O)N1C[C@H](N)C[C@H](C(F)(F)F)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.46
CHRNA3 P32297 4/20 0.46
CHRNA4 P43681 4/20 0.46
CHRNB3 Q05901 2/20 0.46
CHRNA6 Q15825 2/20 0.46
CHRNB4 P30926 2/20 0.42
CHRNA7 P36544 2/20 0.42
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC9A1 P19634 1/20 0.34
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 1/20 0.33
JAK1 P23458 1/20 0.32
JAK3 P52333 1/20 0.32
EPHX2 P34913 1/20 0.30
TACR1 P25103 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27410286 0.81 CHRNB2 (0.41) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL6523733 0.80 SPR (0.32)
SCHEMBL3403409 0.78
SCHEMBL23866581 0.77 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL21661510 0.77 CHRNB2 (0.46) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL10310052 0.75 SPR (0.43) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL15298466 0.71 CHRNB2 (0.53) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL22802776 0.70 CHRNB2 (0.55) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL29348155 0.70 TLR8 (0.30)
SCHEMBL12510683 0.70 EPHX2 (0.47) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020025517-A1 TLR7/8 ANTAGONISTS AND USES THEREOF MERCK PATENT GMBH (DE) 2020-02-06 WO disclosed