SCHEMBL21664047

SCHEMBL21664047

CN1CCN(C(c2ccccn2)c2ccccn2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 6/20 0.64
SLC1A3 P43003 1/20 0.59
BAX Q07812 1/20 0.57
MAPT P10636 3/20 0.56
HTT P42858 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
HSP90AA1 P07900 1/20 0.56
PPP1CA P62136 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
OPRM1 P35372 2/20 0.55
CHRM2 P08172 2/20 0.55
ADRA2A P08913 2/20 0.55
CHRM1 P11229 2/20 0.55
DRD1 P21728 2/20 0.55
DRD3 P35462 2/20 0.55
SLC6A3 Q01959 2/20 0.55
KCNH2 Q12809 2/20 0.55
CHRM4 P08173 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5556390 1.00 IDH1 (0.64) IDH1SLC1A3BAXMAPTHTT
SCHEMBL29504706 0.84 MC4R (0.56) IDH1SLC1A3BAXMAPTHTT
SCHEMBL8305070 0.81 KCNA5 (0.76) IDH1MAPTHTTKDM4EALDH1A1
SCHEMBL11819962 0.79 IDH1 (0.48) IDH1SLC1A3BAXMAPTHTT
SCHEMBL16182262 0.79 IDH1 (0.48) IDH1SLC1A3BAXMAPTHTT
SCHEMBL8304948 0.79 MEN1 (0.55) IDH1MAPTKDM4EALDH1A1LMNA
SCHEMBL9959870 0.78 ALOX12 (0.76) IDH1MAPTHTTKDM4EALDH1A1
SCHEMBL3637549 0.78 IDH1 (0.50) IDH1SLC1A3BAXMAPTHTT
SCHEMBL11813355 0.77 IDH1 (0.49) IDH1SLC1A3BAXMAPTHTT
SCHEMBL30499312 0.77 IDH1 (0.49) IDH1SLC1A3BAXMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3297992-B1 HETEROCYCLICALKYL DERIVATIVE COMPOUNDS AS SELECTIVE HISTONE DEACETYLASE INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2020-02-05 EP disclosed