SCHEMBL2166780

SCHEMBL2166780

COc1c(F)c(F)cc(C(=O)OCCCCO)c1F.CS(=O)(=O)O

nearest known ligand 0.39

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 2/20 0.36
SLC29A1 Q99808 1/20 0.34
CYP3A4 P08684 2/20 0.34
TSHR P16473 2/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2D6 P10635 1/20 0.34
THPO P40225 1/20 0.34
MTOR P42345 1/20 0.34
SCN1A P35498 1/20 0.33
SCN2A Q99250 1/20 0.33
SCN3A Q9NY46 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
PMP22 Q01453 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2166677 0.91 KMT2A (0.35) KMT2AGAAMEN1TSHRALDH1A1
SCHEMBL2168217 0.91 KMT2A (0.36) KMT2AGAAMEN1SLC29A1CYP3A4
SCHEMBL2831392 0.88 KMT2A (0.47) KMT2AGAAMEN1SLC29A1CYP3A4
SCHEMBL2834707 0.86 KMT2A (0.51) KMT2AGAAMEN1SLC29A1CYP3A4
1,4-Butanediol SCHEMBL2166784 0.85 FABP4 (0.36) KMT2AMEN1MAPK1ALDH1A1
SCHEMBL2829961 0.83 KMT2A (0.42) KMT2AGAASLC29A1TSHRSCN1A
SCHEMBL2166953 0.82 KMT2A (0.33) KMT2AGAAMEN1TSHRALDH1A1
SCHEMBL2165984 0.81 GAA (0.34) GAATSHRLMNA
SCHEMBL2170072 0.80 GAA (0.33) GAATSHRLMNA
Ethylene Glycol SCHEMBL2166684 0.79 FABP4 (0.38) KMT2AMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383274-B2 Nonaqueous electrolyte solution for lithium battery, lithium battery using same, and formyloxy group-containing compound used therein UBE INDUSTRIES, LTD. (JP) 2013-02-26 US disclosed
US-20110183199-A1 NONAQUEOUS ELECTROLYTE SOLUTION FOR LITHIUM BATTERY, LITHIUM BATTERY USING SAME, AND FORMYLOXY GROUP-CONTAINING COMPOUND USED THEREIN UBE INDUSTRIES, LTD. (JP) 2011-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183199-A1 NONAQUEOUS ELECTROLYTE SOLUTION FOR LITHIUM BATTERY, LITHIUM BATTERY USING SAME, AND FORMYLOXY GROUP-CONTAINING COMPOUND USED THEREIN HCN2, KCNN2, KCNB1 KMT2A 2361/4885GAA 4111/4885MEN1 2002/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.