SCHEMBL21676745

SCHEMBL21676745

Cn1c(=O)c2ccncc2n1C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 4/20 0.43
NFATC1 O95644 3/20 0.43
GSK3B P49841 3/20 0.43
KDM5A P29375 1/20 0.43
ADORA3 P0DMS8 3/20 0.41
ADORA2A P29274 3/20 0.41
ADORA1 P30542 2/20 0.41
KDM4C Q9H3R0 3/20 0.38
KDM4A O75164 1/20 0.38
KDM4B O94953 1/20 0.38
KDM5C P41229 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
KDM3A Q9Y4C1 1/20 0.38
DAO P14920 1/20 0.37
PLK1 P53350 1/20 0.36
GABRA5 P31644 1/20 0.36
AAK1 Q2M2I8 1/20 0.35
FEN1 P39748 1/20 0.35
KAT2B Q92831 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21676746 0.84 MAOA (0.39) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL23471340 0.80 DYRK1A (0.42) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL13819107 0.77 ADORA3 (0.53) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL16542214 0.72 KDM4C (0.34) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL16542255 0.72 G6PD (0.40) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL22016877 0.72 ADORA3 (0.41) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL1609661 0.72 ADORA3 (0.54) DYRK1ANFATC1GSK3BADORA3ADORA2A
SCHEMBL22016239 0.71 ADORA3 (0.43) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL15624106 0.71 MAPT (0.40) DYRK1ANFATC1GSK3BKDM5AADORA3
SCHEMBL2537047 0.70 ERCC1 (0.52) FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020024997-A1 PREPARATION AND APPLICATION OF CLASS OF N-CONTAINING HETEROCYCLIC COMPOUNDS HAVING IMMUNOREGULATORY FUNCTION 上海轶诺药业有限公司 2020-02-06 WO disclosed