SCHEMBL2167968

SCHEMBL2167968

CC(C)(C)[Si](C)(C)O[C@H]1CC(=O)O[C@H](CI)C1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
BUB1 O43683 1/20 0.32
TOP2A P11388 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595118 1.00 HMGCR (0.36) HMGCRHDAC1HDAC2HDAC6BUB1
SCHEMBL2169371 1.00 HMGCR (0.36) HMGCRHDAC1HDAC2HDAC6BUB1
SCHEMBL10024055 0.87 HMGCR (0.37) HMGCRHDAC1HDAC2HDAC6BUB1
SCHEMBL2168815 0.85 HMGCR (0.36) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL9269812 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL4643619 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL2067039 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL10024054 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL10024025 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A
SCHEMBL4440967 0.85 HMGCR (0.38) HMGCRHDAC1HDAC2HDAC6TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604483-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE 4-HYDROXYTETRAHYDRO-2-PYRANONE DERIVATIVES ZENECA LIMITED (GB) 1994-07-06 EP claimed
WO-1993006235-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE 4-HYDROXYTETRAHYDRO-2-PYRANONE DERIVATIVES ZENECA LIMITED (GB) 1993-04-01 WO claimed
EP-2134696-B1 PROCESSES FOR THE PREPARATION OF STATINS, PARTICULARLY ROSUVASTATIN, AND INTERMEDIATES FOR THE PREPARATION THEREOF LEK PHARMACEUTICALS (SI) 2017-05-17 EP disclosed
EP-2341054-B1 Process for the synthesis of HMG-CoA reductase inhibitors LEK PHARMACEUTICALS (SI) 2014-06-25 EP disclosed
EP-2557084-B1 ROSUVASTATIN CALCIUM INTERMEDIATE AND PREPARATION METHOD THEREOF PORTON FINE CHEMICALS LTD (CN) 2014-06-18 EP disclosed
US-8471045-B2 Synthesis of statins LEK PHARMACEUTICALS D.D. (SI) 2013-06-25 US disclosed
EP-1937696-B1 PROCESS FOR THE SYNTHESIS OF HMG-CoA REDUCTASE INHIBITORS LEK PHARMACEUTICALS (SI) 2013-05-22 EP disclosed
EP-1937696-B1 PROCESS FOR THE SYNTHESIS OF HMG-CoA REDUCTASE INHIBITORS LEK PHARMACEUTICALS (SI) 2013-05-22 EP disclosed
US-8269001-B2 Process for the synthesis of HMG-CoA reductase inhibitors LEK PHARMACEUTICALS D.D. (SI) 2012-09-18 US disclosed
US-8269001-B2 Process for the synthesis of HMG-CoA reductase inhibitors LEK PHARMACEUTICALS D.D. (SI) 2012-09-18 US disclosed
US-20120196333-A1 SYNTHESIS OF STATINS LEK PHARMACEUTICALS D.D. (SI) 2012-08-02 US disclosed
US-20080300406-A1 Process for the Synthesis of Hmg-Coa Reductase Inhibitors LEK PHARMACEUTICALS D.D. (SI) 2008-12-04 US disclosed
US-20080300406-A1 Process for the Synthesis of Hmg-Coa Reductase Inhibitors LEK PHARMACEUTICALS D.D. (SI) 2008-12-04 US disclosed
EP-1978020-A1 Processes for the preparation of statins, particularly rosuvastatin, and intermediates for the preparation thereof LEK Pharmaceuticals D.D. (SI) 2008-10-08 EP disclosed
EP-1937696-A1 PROCESS FOR THE SYNTHESIS OF HMG-CoA REDUCTASE INHIBITORS LEK Pharmaceuticals D.D. (SI) 2008-07-02 EP disclosed
EP-1775299-A1 Process for the synthesis of HMG-CoA reductase inhibitors LEK Pharmaceuticals D.D. (SI) 2007-04-18 EP disclosed
WO-2007039287-A1 PROCESS FOR THE SYNTHESIS OF HMG-CoA REDUCTASE INHIBITORS LEK PHARMACEUTICALS D.D. (SI) 2007-04-12 WO disclosed
US-5443970-A SEPARATION OF ISOMERS IN A MIXTURE BY SELECTIVE REACTION ZENECA LIMITED (GB) 1995-08-22 US disclosed
EP-0604483-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE 4-HYDROXYTETRAHYDRO-2-PYRANONE DERIVATIVES ZENECA LIMITED (GB) 1994-07-06 EP disclosed
WO-1993006235-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY PURE 4-HYDROXYTETRAHYDRO-2-PYRANONE DERIVATIVES ZENECA LIMITED (GB) 1993-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120196333-A1 SYNTHESIS OF STATINS HMGCR, DHCR7, COASY HMGCR 1/4885HDAC1 1079/4885HDAC2 784/4885
US-20080300406-A1 Process for the Synthesis of Hmg-Coa Reductase Inhibitors HMGCR, COASY, LSS HMGCR 1/4885HDAC1 1849/4885HDAC2 1736/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.