SCHEMBL2168920

SCHEMBL2168920

O=C(Cc1nn[nH]n1)NC1CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 1/20 0.62
KDM4A O75164 1/20 0.62
KDM5A P29375 1/20 0.62
ALDH1A1 P00352 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
EPHX1 P07099 1/20 0.45
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
RORC P51449 1/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353804 0.77 KDM6B (0.68) KDM6BKDM4AKDM5AALDH1A1L3MBTL1
SCHEMBL12432401 0.75 KDM6B (0.51) KDM6BKDM4AKDM5AALDH1A1L3MBTL1
SCHEMBL3640002 0.75 CCR5 (0.50)
SCHEMBL18378770 0.74 ENPP2 (0.51) KDM6BKDM4AKDM5AALDH1A1GRIN2D
SCHEMBL18368147 0.72 ENPP2 (0.48) KDM5AALDH1A1GRIN2DGRIN3BGRIN1
SCHEMBL241024 0.71
SCHEMBL5591576 0.70
SCHEMBL19268378 0.69 CA12 (0.69) KDM6BKDM4AKDM5AALDH1A1L3MBTL1
SCHEMBL18116301 0.64 KDM6B (0.51) KDM6BKDM4AKDM5AALDH1A1L3MBTL1
SCHEMBL22576347 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4726238-B2 2011-07-20 JP claimed
EP-1660492-A1 BENZIMIDAZOLE, BENZTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND THEIR USE AS LTA4H MODULATORS Janssen Pharmaceutica N.V. (BE) 2006-05-31 EP claimed
WO-2005012297-A1 BENZIMIDAZOLE, BENZTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND THEIR USE AS LTA4H MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-10 WO claimed