SCHEMBL2170203

SCHEMBL2170203

CS(=O)(=O)[C@]1(COc2ccc(C(F)(F)F)cc2C(N)=O)CCCN1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
PTGDR2 Q9Y5Y4 6/20 0.37
SCN8A Q9UQD0 4/20 0.36
SCN10A Q9Y5Y9 4/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
IRAK4 Q9NWZ3 2/20 0.34
MRGPRX4 Q96LA9 1/20 0.33
MGLL Q99685 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC6A9 P48067 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1974222 0.83 PARP1 (0.45) PARP1PTGDR2SCN8ASCN10ACYP1A2
SCHEMBL2170923 0.81 PARP1 (0.42) PARP1PTGDR2SCN8ASCN10ACYP1A2
SCHEMBL2171049 0.78 PARP1 (0.39) PARP1PTGDR2SCN8ASCN10ACYP1A2
SCHEMBL17180898 0.72 PTGDR2 (0.41) PTGDR2SCN8ASCN10ACYP1A2CYP2C9
SCHEMBL4639880 0.70 CYP1A2 (0.50) PTGDR2SCN8ASCN10ACYP1A2CYP2C9
SCHEMBL3711919 0.69 MRGPRX4 (0.44) PARP1PTGDR2SCN8ASCN10ACYP1A2
SCHEMBL2170206 0.69 CNR2 (0.55) SLC6A9
SCHEMBL2170200 0.69 CNR2 (0.55) SLC6A9
SCHEMBL2171083 0.69 PARP1 (0.38) PARP1PTGDR2SCN8ASCN10AMRGPRX4
SCHEMBL18963341 0.68 CNR2 (0.49) CYP1A2CYP2C9CYP2C19MRGPRX4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346843-A2 SUBSTITUTED BENZAMIDES AS CANNABINOID RECEPTOR LIGANDS Abbott Laboratories (US) 2011-07-27 EP claimed
WO-2010028338-A2 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2010-03-11 WO claimed