SCHEMBL2170923

SCHEMBL2170923

C[C@@]1(COc2ccc(C(F)(F)F)cc2C(N)=O)CCCCN1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.42
SCN8A Q9UQD0 4/20 0.39
SCN10A Q9Y5Y9 4/20 0.39
IRAK4 Q9NWZ3 5/20 0.36
CNR2 P34972 1/20 0.35
TACR1 P25103 3/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1974222 0.97 PARP1 (0.45) PARP1SCN8ASCN10AIRAK4CNR2
SCHEMBL2170203 0.81 PARP1 (0.41) PARP1SCN8ASCN10AIRAK4MRGPRX4
SCHEMBL2171017 0.78 SLC6A4 (0.39) PARP1IRAK4PTGDR2
SCHEMBL2171049 0.78 PARP1 (0.39) PARP1SCN8ASCN10AIRAK4CNR2
SCHEMBL2170542 0.74 LTA4H (0.55) SCN8ASCN10AIRAK4CNR2CYP1A2
SCHEMBL18963341 0.73 CNR2 (0.49) CNR2MRGPRX4CYP1A2CYP2C9CYP2C19
SCHEMBL2169515 0.73 CNR2 (0.51) SCN8ASCN10AIRAK4CNR2CYP1A2
SCHEMBL2171677 0.73 CNR2 (0.51) SCN8ASCN10AIRAK4CNR2CYP1A2
SCHEMBL4639880 0.72 CYP1A2 (0.50) SCN8ASCN10AMRGPRX4CYP1A2CYP2C9
SCHEMBL3711919 0.71 MRGPRX4 (0.44) PARP1SCN8ASCN10AMRGPRX4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346843-A2 SUBSTITUTED BENZAMIDES AS CANNABINOID RECEPTOR LIGANDS Abbott Laboratories (US) 2011-07-27 EP claimed
WO-2010028338-A2 NOVEL COMPOUNDS AS CANNABINOID RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2010-03-11 WO claimed