SCHEMBL21708464

SCHEMBL21708464

CCCC(F)OC(=O)CCC(CN)c1cccc(F)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGFR P43088 3/20 0.35
ALDH1A1 P00352 2/20 0.31
TDP1 Q9NUW8 2/20 0.31
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
ALOX15 P16050 1/20 0.31
MC4R P32245 1/20 0.30
KDM4E B2RXH2 1/20 0.30
TSHR P16473 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708658 0.89 TAS1R3 (0.34) PTGFRALDH1A1MC4RTAS1R3TAS1R1
SCHEMBL21708509 0.85 NISCH (0.36) PTGFRALDH1A1KDM4EL3MBTL1TAS1R3
SCHEMBL21708613 0.85 TAS1R3 (0.33) PTGFRTAS1R3TAS1R1
SCHEMBL21708770 0.84 PTGFR (0.35) PTGFRALDH1A1KDM4EL3MBTL1
Hydrochloric Acid SCHEMBL21708570 0.84 NISCH (0.35) PTGFRALDH1A1KDM4EL3MBTL1TAS1R3
SCHEMBL21708507 0.84 PTGFR (0.33) PTGFR
SCHEMBL21708537 0.82 PTGFR (0.33) PTGFRMC4RL3MBTL1
SCHEMBL21708612 0.81 TAS1R3 (0.32) L3MBTL1TAS1R3TAS1R1
SCHEMBL21708785 0.81 ROCK2 (0.32) PTGFRALDH1A1L3MBTL1
SCHEMBL21708590 0.81 L3MBTL1 (0.41) TDP1KDM4ETSHRL3MBTL1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609870-A1 SUBSTITUTED N-ARYLETHYL-2-AMINOQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed