SCHEMBL21708652

SCHEMBL21708652

CCCC(F)OC(=O)CC(C)(CN)c1ccccc1F

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KCNN4 O15554 5/20 0.33
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
KCNE1 P15382 1/20 0.31
KCNQ1 P51787 1/20 0.31
PRSS1 P07477 1/20 0.30
CTSG P08311 1/20 0.30
CTRB1 P17538 1/20 0.30
CMA1 P23946 1/20 0.30
RIPK1 Q13546 1/20 0.30
KIF11 P52732 1/20 0.30
GPR88 Q9GZN0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708704 0.88 TAS1R3 (0.33) TAS1R3TAS1R1KIF11
SCHEMBL21708743 0.87 MEN1 (0.41) TAS1R3TAS1R1
SCHEMBL21708725 0.81 SMN1; SMN2 (0.35)
SCHEMBL21708656 0.81 TAS1R3 (0.35) TAS1R3TAS1R1
SCHEMBL21708782 0.80 SMN1; SMN2 (0.36) HDAC6ADRB3
SCHEMBL21708772 0.80 PTGFR (0.34) TAS1R3TAS1R1
Hydrochloric Acid SCHEMBL21708639 0.79 PTGFR (0.33)
Hydrochloric Acid SCHEMBL21708672 0.79 NR3C1 (0.36) TAS1R3TAS1R1
SCHEMBL21656595 0.78 KCNN4 (0.39) HDAC3HDAC1HDAC2HDAC6KCNN4
SCHEMBL21631996 0.74 CYP2C19 (0.53) HDAC3HDAC1HDAC2HDAC6KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed