SCHEMBL21708663

SCHEMBL21708663

CCCC(F)OC(=O)C(CN)c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.44
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KCNQ2 O43526 1/20 0.38
AOC3 Q16853 1/20 0.38
CASR P41180 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
EPHX1 P07099 4/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708758 0.86 ROCK2 (0.45) ROCK2ALDH1A1KCNQ2AOC3MAPK1
SCHEMBL21708677 0.84 ROCK2 (0.49) ROCK2KCNQ2AOC3CASRMAPK1
SCHEMBL21708787 0.81 HPGD (0.39) MEN1KMT2AALDH1A1CASRCYP1A2
SCHEMBL21656358 0.76 MEN1 (0.44) ROCK2MEN1KMT2AMAPTNPC1
SCHEMBL21708777 0.73 KMT2A (0.38) MEN1KMT2AMAPTNPC1ALDH1A1
SCHEMBL19612687 0.73 MEN1 (0.49) MEN1KMT2AALDH1A1NPSR1KCNQ2
SCHEMBL5820507 0.73 MEN1 (0.60) MEN1KMT2AALDH1A1NPSR1KCNQ2
SCHEMBL6985765 0.72 MEN1 (0.63) ROCK2MEN1KMT2AALDH1A1NPSR1
SCHEMBL6983317 0.72 MEN1 (0.63) ROCK2MEN1KMT2AALDH1A1NPSR1
SCHEMBL6976406 0.72 MEN1 (0.63) ROCK2MEN1KMT2AALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed