SCHEMBL21708787

SCHEMBL21708787

CCCC(F)OC(=O)CC(CN)c1cccc(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CASR P41180 1/20 0.38
GABBR2 O75899 4/20 0.37
GABBR1 Q9UBS5 4/20 0.37
LMNA P02545 2/20 0.37
CYP2C9 P11712 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP3A4 P08684 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
NFKB1 P19838 1/20 0.37
DRD3 P35462 1/20 0.37
BLM P54132 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
THRB P10828 1/20 0.37
TSHR P16473 1/20 0.37
EPHX1 P07099 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708683 0.87 F10 (0.38) GABBR2GABBR1CYP2C9CYP3A4CYP1A2
SCHEMBL21708681 0.85 L3MBTL1 (0.46) CASR
SCHEMBL21708792 0.82 TAS1R3 (0.33) GABBR2GABBR1LMNACYP2C9MEN1
SCHEMBL21708663 0.81 ROCK2 (0.44) HPGDALDH1A1CASRCYP2C9MEN1
SCHEMBL21708777 0.81 KMT2A (0.38) HPGDALDH1A1CASRMEN1KMT2A
SCHEMBL563435 0.80 F10 (0.48) HPGDALDH1A1GABBR2GABBR1LMNA
SCHEMBL21609293 0.80 F2 (0.47) HPGDALDH1A1GABBR2GABBR1LMNA
SCHEMBL29848001 0.80 F2 (0.47) HPGDALDH1A1GABBR2GABBR1LMNA
SCHEMBL21708638 0.79 GABBR2 (0.38) ALDH1A1GABBR2GABBR1LMNACYP2C9
SCHEMBL21708646 0.79 NISCH (0.37) HPGDALDH1A1GABBR2GABBR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed