SCHEMBL21708682

SCHEMBL21708682

CCCC(F)OC(=O)CCCC(C#N)c1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 4/20 0.39
CASP1 P29466 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
CYSLTR2 Q9NS75 1/20 0.33
CYSLTR1 Q9Y271 1/20 0.33
PPARG P37231 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
NPSR1 Q6W5P4 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HPGD P15428 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
RECQL P46063 1/20 0.31
LMNA P02545 2/20 0.31
GLS O94925 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708512 0.93 CCR1 (0.36) CCR1CASP1L3MBTL1TAS1R3TAS1R1
SCHEMBL21708675 0.87 CCR1 (0.37) CCR1CASP1TAS1R3TAS1R1NPSR1
SCHEMBL21708716 0.81 L3MBTL1 (0.36) CASP1L3MBTL1CYSLTR2CYSLTR1PPARG
SCHEMBL21708707 0.81 CCR1 (0.36) CCR1TAS1R3TAS1R1NPSR1MEN1
SCHEMBL21708518 0.81 TAS1R3 (0.32) L3MBTL1TAS1R3TAS1R1MEN1KMT2A
SCHEMBL21708548 0.81 MEN1 (0.35) CYSLTR2CYSLTR1NPSR1MEN1KMT2A
SCHEMBL21708569 0.80 KMT2A (0.33) L3MBTL1KMT2A
SCHEMBL21708544 0.80 POLB (0.38) L3MBTL1PPARGTAS1R3TAS1R1NPSR1
SCHEMBL21656588 0.79 CCR1 (0.42) CCR1CASP1ALDH1A1GLS
SCHEMBL21632085 0.78 CCR1 (0.48) CCR1CYSLTR2CYSLTR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed