SCHEMBL21708707

SCHEMBL21708707

CCCC(F)OC(=O)CCC(C#N)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
CYP3A4 P08684 1/20 0.32
KDM4E B2RXH2 1/20 0.32
EEF2K O00418 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
MC4R P32245 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708459 0.89 CCR1 (0.32) CCR1LMNAKMT2AADRB1
SCHEMBL21708548 0.88 MEN1 (0.35) ALDH1A1LMNAMEN1KMT2ANPSR1
SCHEMBL21708512 0.87 CCR1 (0.36) CCR1TAS1R3TAS1R1ALDH1A1LMNA
SCHEMBL21708544 0.87 POLB (0.38) TAS1R3TAS1R1LMNAMEN1KMT2A
SCHEMBL21708545 0.87 KMT2A (0.33) TAS1R3TAS1R1KMT2AADRB2ADRB1
SCHEMBL21708482 0.86 CES2 (0.33) KMT2ACES2CES1
SCHEMBL21708654 0.85 MEN1 (0.38) LMNAMEN1KMT2AKDM4E
SCHEMBL21708473 0.85 CNR2 (0.34) ALDH1A1KMT2ACYP3A4KDM4ECNR2
SCHEMBL21708466 0.83 F2R (0.36)
SCHEMBL21708737 0.81 CES2 (0.33) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed