SCHEMBL21708941

SCHEMBL21708941

C#CCOc1ccc2c(c1)c(CCN)cn2CC#C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.46
EGFR P00533 7/20 0.44
IGF1R P08069 7/20 0.44
FLT4 P35916 7/20 0.44
KDR P35968 7/20 0.44
HTR6 P50406 4/20 0.38
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HTR1D P28221 3/20 0.36
HTR1A P08908 2/20 0.36
HTR1B P28222 2/20 0.36
MTNR1A P48039 2/20 0.35
CASR P41180 1/20 0.35
MAOA P21397 1/20 0.35
ACHE P22303 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708936 0.83 HTR6 (0.42) EGFRIGF1RFLT4KDRHTR6
SCHEMBL21693977 0.83 MTNR1A (0.42) ADRB2HTR6POLBMAPTNPSR1
Hydrochloric Acid SCHEMBL21693927 0.82 MTNR1A (0.41) ADRB2EGFRIGF1RFLT4KDR
SCHEMBL21709087 0.79 EGFR (0.42) ADRB2EGFRIGF1RFLT4KDR
Hydrochloric Acid SCHEMBL21693918 0.78 EGFR (0.43) ADRB2EGFRIGF1RFLT4KDR
SCHEMBL8758848 0.76 HTR2A (0.55) HTR6POLBMAPT
SCHEMBL21709108 0.75 HTR6 (0.38) EGFRIGF1RFLT4KDRHTR6
SCHEMBL12790242 0.74 HTR6 (0.55) ADRB2EGFRIGF1RFLT4KDR
SCHEMBL12790246 0.72 HTR6 (0.57) ADRB2EGFRIGF1RFLT4KDR
SCHEMBL14801810 0.72 CHEK1 (0.37) ADRB2HTR6POLBHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed