SCHEMBL21709108

SCHEMBL21709108

C#CCOc1ccc2c(c1)c(CCN(CC#C)C(=O)C(F)(F)F)cn2CC#C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 5/20 0.38
LTB4R Q15722 2/20 0.35
LTB4R2 Q9NPC1 2/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MTNR1A P48039 4/20 0.34
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
PPARG P37231 1/20 0.33
KCNH2 Q12809 1/20 0.32
MTNR1B P49286 1/20 0.31
PLA2G4A P47712 1/20 0.31
PLA2G2A P14555 1/20 0.31
EGFR P00533 2/20 0.31
IGF1R P08069 2/20 0.31
FLT4 P35916 2/20 0.31
KDR P35968 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708936 0.82 HTR6 (0.42) HTR6LTB4RLTB4R2POLBMAPT
SCHEMBL21708941 0.75 ADRB2 (0.46) HTR6POLBMAPTNPSR1MTNR1A
SCHEMBL21693977 0.72 MTNR1A (0.42) HTR6POLBMAPTNPSR1MTNR1A
Hydrochloric Acid SCHEMBL21693927 0.71 MTNR1A (0.41) HTR6POLBMAPTNPSR1MTNR1A
SCHEMBL21708905 0.67 HTR6 (0.39) HTR6MAPTMAOAMAOBPLA2G2A
SCHEMBL17469273 0.61 POLB (0.46) POLBMAPTNPSR1MTNR1AMAOA
SCHEMBL16629671 0.61 CYP19A1 (0.47) EGFRIGF1RFLT4KDR
SCHEMBL21709087 0.59 EGFR (0.42) HTR6MAPTNPSR1PLA2G2AEGFR
SCHEMBL24733324 0.58 PLOD2 (0.55)
Hydrochloric Acid SCHEMBL21693918 0.58 EGFR (0.43) HTR6MAPTNPSR1PLA2G2AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed