SCHEMBL21709062

SCHEMBL21709062

C#CCOc1cc(CCN(CC#C)CC#C)ccc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA4 P22748 1/20 0.46
CA9 Q16790 1/20 0.46
DRD3 P35462 3/20 0.43
TSHR P16473 2/20 0.43
DRD1 P21728 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.43
NFKB1 P19838 1/20 0.43
DRD4 P21917 1/20 0.43
DRD5 P21918 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709061 0.87 CA12 (0.46) CA12CA1CA2CA4CA9
SCHEMBL21709064 0.81 TAAR1 (0.58) DRD3TSHRDRD1CYP3A4CYP2D6
SCHEMBL21709160 0.78 CA12 (0.35) CA12CA1CA2CA4CA9
SCHEMBL21708854 0.76 CGAS (0.33) CA12CA1CA2CA4CA9
SCHEMBL21709060 0.75 ACHE (0.43) DRD3TSHRDRD1DRD2NFKB1
SCHEMBL21709156 0.74 BCHE (0.36) CA12CA1CA2CA4CA9
SCHEMBL21709075 0.74 CYP1A2 (0.61) CA2CYP3A4CYP2D6KDM4EPMP22
SCHEMBL21709057 0.73 CYP3A4 (0.40) TSHRDRD1CYP3A4CYP2D6DRD2
SCHEMBL23784797 0.70 CALM1 (0.53) TSHRTAAR1MAPK1PTPN1
SCHEMBL7688903 0.69 KDM4E (0.53) TSHRDRD2KDM4ETAAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed