SCHEMBL21709097

SCHEMBL21709097

C#CCN(CC#C)CCc1c[nH]c2cc(C#C)c(O)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 6/20 0.45
HTR2A P28223 8/20 0.42
HTR2C P28335 6/20 0.42
HTR2B P41595 4/20 0.42
HTR1A P08908 7/20 0.40
SLC6A4 P31645 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR6 P50406 4/20 0.38
MPO P05164 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
HTR1E P28566 3/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
SLC6A2 P23975 2/20 0.36
ADRA1A P35348 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709103 0.80 HTR2C (0.57) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL25057123 0.79 HTR1D (0.71) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL21709105 0.77 HTR1D (0.42) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL21709102 0.77 KDM4E (0.42) HTR1DHTR2AHTR2CSLC6A4CYP1A2
SCHEMBL26989208 0.75 HTR1A (0.66) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL21709150 0.73 CA12 (0.39) HTR1ACYP2D6HSD17B10ADRA1AADRA1B
SCHEMBL21709101 0.72 HTR1A (0.46) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL25057107 0.70 HTR1D (0.55) HTR1DHTR2AHTR2CHTR2BHTR1A
SCHEMBL21708880 0.65 CA12 (0.43) CYP2D6HSD17B10ADRA1AADRA1BDRD3
SCHEMBL21708854 0.65 CGAS (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed