SCHEMBL21709150

SCHEMBL21709150

C#CCN(CC#C)CCc1cc(O)c(O)cc1C#C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
HTR1A P08908 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
DRD2 P14416 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
DRD3 P35462 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708854 0.83 CGAS (0.33) CA12CA1CA2CA4CA9
SCHEMBL21709269 0.76 BCHE (0.39) CA12CA1CA2CA4CA9
SCHEMBL21708853 0.75 BCHE (0.36) CA12CA1CA2CA4CA9
SCHEMBL21708880 0.74 CA12 (0.43) CA12CA1CA2CA4CA9
SCHEMBL21709097 0.73 HTR1D (0.45) HTR1ACYP2D6DRD2ADRA1DADRA1A
SCHEMBL21709141 0.73 TSHR (0.35) CA12CA1CA2CA4CA9
SCHEMBL21709190 0.73 HMGCR (0.40) CYP3A4CYP2D6DRD2TSHRNFKB1
SCHEMBL21709105 0.70 HTR1D (0.42) HTR1ACYP3A4CYP2D6TSHRDRD1
SCHEMBL21709148 0.70 ACHE (0.35) MAOAMAOB
SCHEMBL21709161 0.68 ADRB2 (0.31) CYP3A4ADRA1AHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed