SCHEMBL21709102

SCHEMBL21709102

C#CCNCCc1c[nH]c2cc(C#C)c(O)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
CYP2D6 P10635 3/20 0.42
MEN1 O00255 1/20 0.42
HTR2C P28335 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
HPGD P15428 2/20 0.41
APEX1 P27695 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTR2A P28223 2/20 0.41
MPO P05164 5/20 0.40
SLC6A4 P31645 1/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709103 0.80 HTR2C (0.57) CYP2D6MEN1HTR2CKMT2ANPSR1
SCHEMBL25057132 0.79 HTR2C (0.68) KDM4ECYP2D6MEN1HTR2CKMT2A
SCHEMBL21709097 0.77 HTR1D (0.45) CYP2D6HTR2CCYP1A2HSD17B10HTR2A
SCHEMBL26989205 0.75 HTR2A (0.70) KDM4EMEN1KMT2ACYP1A2HTR2A
SCHEMBL26989142 0.75 MTNR1A (0.60) HTR2CMTNR1AMTNR1BHPGDHTR2A
SCHEMBL29206374 0.74 MPO (0.73) KMT2AMTNR1AMTNR1BHTR2AMPO
SCHEMBL21709148 0.73 ACHE (0.35) HTR2CHTR2AMPO
SCHEMBL21709099 0.72 HTR2A (0.46) KDM4ECYP2D6MEN1HTR2CKMT2A
SCHEMBL31708144 0.71 HTR2A (0.70) KDM4EMEN1HTR2CKMT2ANPSR1
SCHEMBL26989179 0.68 HTR2C (0.63) KDM4ECYP2D6MEN1HTR2CKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed