SCHEMBL21709098

SCHEMBL21709098

C#CCOc1ccc2[nH]cc(CCN)c2c1C#C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 10/20 0.45
HTR2C P28335 5/20 0.42
HTR1D P28221 9/20 0.39
HTR1A P08908 8/20 0.39
HTR1B P28222 8/20 0.39
HTR2B P41595 2/20 0.38
PARP1 P09874 1/20 0.38
TRPM8 Q7Z2W7 4/20 0.36
CYP1A2 P05177 3/20 0.36
HTR7 P34969 3/20 0.36
HTR6 P50406 3/20 0.36
NFKB1 P19838 2/20 0.36
TSHR P16473 2/20 0.36
HTR4 Q13639 2/20 0.36
MAPT P10636 1/20 0.36
MPO P05164 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
TAAR1 Q96RJ0 2/20 0.36
CYP2A6 P11509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709092 0.77 HTR2C (0.57) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL21709104 0.72 HTR1A (0.45) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL25057108 0.71 HTR1A (0.72) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL1971484 0.67 HTR2A (0.67) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL3210741 0.67 HTR2A (0.67) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL2541508 0.66 HTR2A (0.65) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL8549376 0.66 HTR1A (0.55) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL8544820 0.65 HTR1A (0.54) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL8543442 0.65 HTR1A (0.54) HTR2AHTR2CHTR1DHTR1AHTR1B
SCHEMBL21708858 0.64 HTR2A (0.42) HTR2AHTR2CHTR2BTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed