SCHEMBL21709153

SCHEMBL21709153

C#CCOc1cc(CCN)cc(C#C)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.36
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
HTR2A P28223 5/20 0.36
HTR2C P28335 4/20 0.36
HTR2B P41595 4/20 0.36
LMNA P02545 3/20 0.36
GLA P06280 1/20 0.36
TRPV1 Q8NER1 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
NFKB1 P19838 1/20 0.33
MAOB P27338 1/20 0.32
APEX1 P27695 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ATM Q13315 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709157 0.84 HTR2A (0.40) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL21709163 0.81 ACHE (0.37) HTR2ATRPV1
SCHEMBL21709160 0.81 CA12 (0.35) TRPV1
SCHEMBL21709064 0.77 TAAR1 (0.58) TAAR1TSHRMAPK1LMNAGLA
SCHEMBL21708877 0.73 HTR2A (0.39) TAAR1TSHRMAPK1HTR2ALMNA
SCHEMBL21709066 0.73 KDM4E (0.51) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL21709214 0.72
SCHEMBL21708858 0.72 HTR2A (0.42) TAAR1HTR2AHTR2CHTR2BMAOB
SCHEMBL20970882 0.71 HTR2A (0.66) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL6660288 0.69 ATM (0.68) TAAR1TSHRMAPK1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed