SCHEMBL21708877

SCHEMBL21708877

C#CCOc1cc(CCN)c(C#C)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.39
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
RAD52 P43351 2/20 0.36
RECQL P46063 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
APEX1 P27695 2/20 0.36
GAPDH P04406 1/20 0.36
THRB P10828 1/20 0.36
BLM P54132 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
AGO2 Q9UKV8 1/20 0.35
CGAS Q8N884 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708858 0.88 HTR2A (0.42) HTR2AMAOBTAAR1
SCHEMBL21708864 0.81 HTR2A (0.33) HTR2AMAPTCGAS
SCHEMBL21708854 0.81 CGAS (0.33) CGASMAOB
SCHEMBL21708902 0.75 ADRA2A (0.35) MEN1KMT2ARAD52RECQLTDP1
SCHEMBL21709064 0.74 TAAR1 (0.58) MEN1KMT2ARECQLTDP1APEX1
SCHEMBL21709153 0.73 TAAR1 (0.36) HTR2AMEN1KMT2ARECQLTDP1
SCHEMBL21709245 0.72 P2RX3 (0.31) CGAS
SCHEMBL21709091 0.71 TAAR1 (0.53) HTR2ATAAR1
SCHEMBL26011914 0.70 HTR2A (0.61) HTR2ATAAR1
SCHEMBL21709157 0.69 HTR2A (0.40) HTR2AKDM4EMAPK1TSHRMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed