SCHEMBL21709157

SCHEMBL21709157

C#CCOc1cc(CCN)cc(C#C)c1OCC#C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.40
HTR2C P28335 4/20 0.40
HTR2B P41595 4/20 0.40
MAOB P27338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ATM Q13315 1/20 0.33
TAAR1 Q96RJ0 2/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GSTP1 P09211 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
LOXL2 Q9Y4K0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709153 0.84 TAAR1 (0.36) HTR2AHTR2CHTR2BMAOBKDM4E
SCHEMBL21709156 0.80 BCHE (0.36)
SCHEMBL20970882 0.78 HTR2A (0.66) HTR2AHTR2CHTR2BKDM4EATM
SCHEMBL21709090 0.75 HTR2A (0.69) HTR2AHTR2CHTR2BKDM4EATM
SCHEMBL21709066 0.74 KDM4E (0.51) HTR2AHTR2CHTR2BMAOBKDM4E
SCHEMBL21708858 0.73 HTR2A (0.42) HTR2AHTR2CHTR2BMAOBTAAR1
SCHEMBL21709155 0.72 NFKB1 (0.35) MAOBKDM4ETAAR1TSHRMAPK1
SCHEMBL21709064 0.72 TAAR1 (0.58) KDM4EATMTAAR1TSHRMAPK1
SCHEMBL21709213 0.71 MAOB (0.30) MAOB
SCHEMBL6660288 0.70 ATM (0.68) HTR2AHTR2CHTR2BMAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed