SCHEMBL21709155

SCHEMBL21709155

C#CCOc1cc(C(O)CN)cc(C#C)c1OCC#C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.35
BLM P54132 3/20 0.35
PMP22 Q01453 1/20 0.35
MAOB P27338 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
TAAR1 Q96RJ0 3/20 0.31
MAPT P10636 2/20 0.31
HPGD P15428 2/20 0.31
APEX1 P27695 2/20 0.31
RECQL P46063 2/20 0.31
TDP1 Q9NUW8 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRA2A P08913 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADRB3 P13945 1/20 0.31
DRD2 P14416 1/20 0.31
ADRA2B P18089 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709213 0.82 MAOB (0.30) MAOB
SCHEMBL21709218 0.82 MAOA (0.31)
SCHEMBL21709145 0.82 KDM1A (0.35) MAOBSMN1; SMN2LMNA
SCHEMBL21709070 0.77 NFKB1 (0.50) NFKB1BLMPMP22MAPTADRA2A
SCHEMBL21708865 0.77 MAOB (0.33) BLMMAOBMAPTHPGDAPEX1
SCHEMBL21708896 0.77 NFKB1 (0.49) NFKB1BLMPMP22MAOBTAAR1
SCHEMBL21709144 0.75 NFKB1 (0.41) NFKB1BLMPMP22MAOBTAAR1
SCHEMBL21709056 0.74 NFKB1 (0.61) NFKB1BLMPMP22MAOBTAAR1
SCHEMBL21708902 0.73 ADRA2A (0.35) NFKB1BLMPMP22MAOBTAAR1
SCHEMBL21709157 0.72 HTR2A (0.40) MAOBSMN1; SMN2TAAR1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed