SCHEMBL2171034

SCHEMBL2171034

COCC(OC(=O)c1cc(-c2ccc(C)cn2)cc(-c2cccc(F)c2F)c1)C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 6/20 0.39
P2RX2 Q9UBL9 6/20 0.39
NR1I2 O75469 2/20 0.39
CTSA P10619 4/20 0.36
HPGDS O60760 1/20 0.35
ADORA2A P29274 1/20 0.34
MET P08581 1/20 0.34
GABRA5 P31644 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
SSTR2 P30874 1/20 0.33
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171503 0.87 P2RX3 (0.43) P2RX3P2RX2NR1I2CTSAHPGDS
SCHEMBL2170986 0.84 NR1I2 (0.45) P2RX3P2RX2NR1I2CTSAHPGDS
SCHEMBL2172000 0.80 S1PR3 (0.40) P2RX3P2RX2
SCHEMBL2171032 0.80 P2RX3 (0.49) P2RX3P2RX2NR1I2CTSA
SCHEMBL2172363 0.80 P2RX3 (0.49) P2RX3P2RX2NR1I2CTSAGABRA5
SCHEMBL2172956 0.78 NR1I2 (0.45) P2RX3P2RX2NR1I2CTSAHPGDS
SCHEMBL2171499 0.74 P2RX3 (0.61) P2RX3P2RX2NR1I2
SCHEMBL7947489 0.73 P2RX3 (0.50) P2RX3P2RX2NR1I2CTSA
SCHEMBL2171711 0.73 CYP3A4 (0.46) P2RX3P2RX2NR1I2HPGDSMET
SCHEMBL2172981 0.72 P2RX3 (0.39) P2RX3P2RX2NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346825-A2 MODULATORS OF P2X3 RECEPTOR ACTIVITY Evotec AG (DE) 2011-07-27 EP disclosed