SCHEMBL2171503

SCHEMBL2171503

Cc1ccc(-c2cc(C(=O)O[C@@H](C)C(N)=O)cc(-c3cccc(F)c3F)c2)nc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 7/20 0.43
P2RX2 Q9UBL9 6/20 0.43
NR1I2 O75469 3/20 0.43
HPGDS O60760 1/20 0.37
CTSA P10619 3/20 0.35
DYRK1A Q13627 1/20 0.35
ADORA2A P29274 1/20 0.35
PTGS2 P35354 1/20 0.34
CYP2C9 P11712 2/20 0.34
MET P08581 1/20 0.34
GABRA5 P31644 1/20 0.34
UGT1A1 P22309 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171034 0.87 P2RX3 (0.39) P2RX3P2RX2NR1I2HPGDSCTSA
SCHEMBL2170986 0.85 NR1I2 (0.45) P2RX3P2RX2NR1I2HPGDSCTSA
SCHEMBL2172981 0.83 P2RX3 (0.39) P2RX3P2RX2NR1I2
SCHEMBL2172956 0.81 NR1I2 (0.45) P2RX3P2RX2NR1I2HPGDSCTSA
SCHEMBL2171685 0.79 S1PR3 (0.42) P2RX3P2RX2NR1I2
SCHEMBL2170462 0.77 S1PR3 (0.41) P2RX3P2RX2NR1I2HPGDS
SCHEMBL2172263 0.77 NSD2 (0.37) P2RX3P2RX2
SCHEMBL2171499 0.77 P2RX3 (0.61) P2RX3P2RX2NR1I2
SCHEMBL2171711 0.76 CYP3A4 (0.46) P2RX3P2RX2NR1I2HPGDSPTGS2
SCHEMBL2187309 0.76 P2RX3 (0.56) P2RX3P2RX2NR1I2CTSACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346825-A2 MODULATORS OF P2X3 RECEPTOR ACTIVITY Evotec AG (DE) 2011-07-27 EP disclosed